※1999年以前の論文はこちらのページからどうぞ。
★は更新した部分です。
2009
★207.
Kazuishi Makino, Sayaka Kubota, Sousuke Hara, Masaru Sakaguchi, Akinari Hamajima, Yasumasa Hamada:
Reagent-controlled diastereoselective synthesis of (2S,3R)- and (2R,3R)-2,3-diaminobutanoic acid derivatives using proline-catalyzed α-hydrazination reaction
Tetrahedron, 65, 9468-9473, (2009)
★206.
Takuya Hibino, Kazuishi Makino, Takaya Sugiyama, Yasumasa Hamada:
Homogeneous Chiral Nickel-Catalyzed Asymmetric Hydrogenation of Substituted Aromatic -Aminoketone Hydrochlorides through Dynamic Kinetic Resolution
ChemCatChem, 1, 237-240, (2009)
★205.
Hang Jiang and Yasumasa Hamada:
Highly enantioselective synthesis of angelmarin
Org. Biomol. Chem., 4173-4176, (2009)
★204.
Tetsuhiro Nemoto, Mutsumi Kanematsu, Shinji Tamura, Yasumasa Hamada:
Palladium-Catalyzed Asymmetric Allylic Alkylation of 2,3-Allenyl Acetates Using a Chiral Diaminophosphine Oxide
Adv. Synth. Catal., 351, 1773-1778, (2009)
★203.
Hiromi Arai, Naomi Sugaya, Neri Sasaki, Kazuishi Makino, Sylvain Lectard, Yasumasa Hamada:
Enantioselective aziridination reaction of α,β-unsaturated aldehydes using an organocatalyst and tert-butyl N-arenesulfonyloxycarbamates
Tetrahedron Lett., 50, 3329-3332, (2009)
★202.
Kazuishi Makino, Takayuki Goto, Junpei Ohtaka, Yasumasa Hamada:
Highly stereoselective synthesis of (2R,3R)-2-amino-3-cyclohexyl-3-hydroxypropionic acid using asymmetric hydrogenation
Heterocycles, 77, 629-634, (2009)
★201.
Masaru Sakaguch, Sousuke Hara, Youhei Koma, Kazuishi Makino, Yasumasa Hamada:
Total synthesis of halipeptin D
Peptide Science , 45th, 183-186, (2009)
2008
★200.
Kazuishi Makino, Takayuki Goto, Yasuhiro Hiroki, Yasumasa Hamada:
Direct anti-selective asymmetric hydrogenation of α-amino-β-keto esters through dynamic kinetic resolution using Ru-axially chiral phosphine catalysts-stereoselective synthesis of anti-β-hydroxy-α-amino acids
Tetrahedron: Asymmetry, 19, 2816-2828, (2008)
★199.
Osamu Hara, Hiroshi Fujino, Kazuishi Makino, Yasumasa Hamada:
Palladium-catalyzed asymmetric intramolecular metallo-ene reaction using monodentate phosphines, 9-PBN and 9-NapBN
Heterocycles, 76, 197-202, (2008)
198.
Yasumasa Hamada, Kazuishi Makino:
Catalytic anti-selective asymmetric hydrogenation of α-amino-β-keto esters through dynamic kinetic resolution
Yuki Gosei Kagaku Kyokaishi, 66, 1057-1065, (2008)
197.
Yu Koseki, Takefumi Fujii, Tsukuru Maeda, Takuya Hibino, Kazuishi Makino, Yasumasa Hamada:
Catalytic asymmetric hydrogenation of α-amino-β-keto ester hydrochlorides using homogeneous chiral nickel-bisphosphine complexes through DKR
Chemical communications, 46, 6206-6208, (2008)
196.
Yayoi Yoshitomi , Hiromi Arai, Kazuishi Makino, Yasumasa Hamada:
Enantioselective synthesis of martinelline chiral core and its diastereomer using asymmetric tandem Michael-aldol reaction
Tetrahedron, 64, 11568-11579, (2008)
195.
Osamu Hara, Hiroshi Fujino, Kazuishi Makino, Yasumasa Hamada:
Palladium-catalyzed asymmetric intramolecular metallo-ene reaction using monodentate phosphines, 9-PBN and 9-NapBN
Heterocycles, 76, 197-202, (2008)
194.
Long Jin, Tetsuhiro Nemoto, Hiroshi Nakamura, Yasumasa Hamada:
Pd-catalyzed asymmetric allylic aminations with aromatic amine nucleophiles using chiral diaminophosphine oxides: DIAPHOXs
Tetrahedron: Asymmetry, 19, 1106-1113. (2008)
193.
Yasumasa Hamada, Kazuishi Makino:
Steroselective synthesis of 3-hydroxyproline derivative using asymmetric aldol reaction
Fain Kemikaru, 37, 39-45. (2008)
192.
Tetsuhiro Nemoto, Shinji Tamura, Tatsurou Sakamoto, Yasumasa Hamada:
Pd-Catalyzed asymmetric allylic aminations with aromatic amine nucleophiles using chiral diaminophosphine oxides: DIAPHOXs
Tetrahedron: Asymmetry, 19, 1751-1759. (2008)
2007
191.
Tetsuhiro Nemoto, Tsukasa Hitomi, Hiroshi Nakamura, Long Jin, Keiichiro Hatano, and Yasumasa Hamada:
Synthesis of novel P-stereogenic phenylphosphonamides and their application to Lewis base-catalyzed asymmetric allylation of benzaldehyde
Tetrahedron: Asymmetry, 18, 1844-1849. (2007)
190.
Tetsuhiro Nemoto, Teisuke Harada, Takayoshi Matsumoto, and Yasumasa Hamada:
Pd-catalyzed enantioselective synthesis of quaternary α-amino acid derivatives using a phenylalanine-derived P-chirogenic diaminophosphine oxide
Tetrahedron Lett., 48, 6304-6307. (2007)
189.
Tetsuhiro Nemoto, Yasumasa Hamada:
Pd-catalyzed asymmetric allylic substitution reactions using P-chirogenic diaminophosphine oxides: DIAPHOXs
The Chemical Record, 7, 150-158. (2007)
188.
Osamu Hara, Tomoaki Koshizawa, Kazuishi Makino, Iyo Kunimune, Atsushi Namiki, Yasumasa Hamada:
Synthesis of 2,6-dimethyl-9-aryl-9-phosphabicyclo[3.3.1]nonanes:
their application to asymmetric synthesis of chiral tetrahydroquinolines and relatives
Tetrahedron, 63, 6170-6181. (2007)
187.
Yayoi Yoshitomi, Kazuishi Makino, Yasumasa Hamada:
Organocatalytic Synthesis of (2S,3R)-3-Hydroxy-3-methyl-proline (OHMePro),
a Component of Polyoxypeptins, and Relatives Using OHMePro Itself as a Catalyst
Organic Lett., 9, 2457-2460. (2007)
186.
Tetsuhiro Nemoto, Tatsurou Sakamoto, Takashi Fukuyama, Yasumasa Hamada:
Ir-catalyzed asymmetric allylic alkylation using chiral diaminophosphine
oxides: DIAPHOXs. Formal enantioselective synthesis of (-)-paroxetine.
Tetrahedron Lett., 48, 4977-4981. (2007)
185.
Tetsuhiro Nemoto, Takashi Fukuyama, Eri Yamamoto, Shinji Tamura, Tomoaki Fukuda, Takayoshi Matsumoto, Yuichi Akimoto, Yasumasa Hamada:
Pd-catalyzed asymmetric allylic amination of Morita-Baylis-Hillman adduct derivatives using chiral diaminophosphine oxides: DIAPHOXs.
Organic Lett., 9, 927-930. (2007)
2006
184.
Sousuke Hara, Eri Nagata, Taeko Fujie, Miyako Fujii, Yousuke Takanashi, Kazuishi Makino, Yasumasa Hamada:
Synthetic studies on papuamides, marine cyclodepsipeptides.
Peptide Science, 43, 64-65. (2006)
183.
Tetsuhiro Nemoto, Tatsurou Sakamoto, Takayoshi Matsumoto and Yasumasa Hamada:
Ir-catalyzed asymmetric allylic amination using chiral diaminophosphine oxides.
Tetrahedron Lett., 47, 8737-8740 (2006).
182.
Kazuishi Makino, Masamichi Iwasaki, and Yasumasa Hamada:
Enantio- and Diastereoselective Hydrogenation via Dynamic Kinetic Resolution
by a Cationic Iridium Complex in the Synthesis of b
-Hydroxy-a-amino Acid Esters.
Organic Lett., 8, 4573-4576 (2006).
181.
Tetsuhiro Nemoto, Long Jin, Hiroshi Nakamura and Yasumasa Hamada:
Pd-catalyzed asymmetric allylic alkylation with nitromethane using a chiral diaminophosphine oxide:
(S,RP)-Ph-DIAPHOX. Enantioselective synthesis of (R)-preclamol and (R)-baclofen.
Tetrahedron Lett., 47, 6577-6581 (2006).
180.
Kazuishi Makino, Hang Jiang, Tatsuya Suzuki and Yasumasa Hamada:
The efficient synthesis of (3R,5R)-5-hydroxypiperazic acid and its diastereomer
using Lewis acid-promoted diastereoselective Strecker synthesis.
Tetrahedron: Asymmetry, 17, 1644-1649 (2006).
179.
Kazuishi Makino, Takefumi Fujii and Yasumasa Hamada:
Rhodium-catalyzed asymmetric hydrogenation through dynamic kinetic resolution:
asymmetric synthesis of anti-b
-hydroxy-a-amino acid esters.
Tetrahedron: Asymmetry, 17, 481-485 (2006).
178.
Tetsuhiro Nemoto, Tomoaki Fukuda, and Yasumasa Hamada: Efficient Synthesis of 3-Substituted
2,3-Dihydroquinolin-4-ones Using a One-pot Sequential Multi-catalytic Process:
Pd-catalyzed Allylic Amination – Thiazolium Salt-catalyzed Stetter Reaction
Cascade. Tetrahedron Lett., 47,4365-4368 (2006).
177.
Sousuke Hara, Kazuishi Makino, and Yasumasa Hamada:Synthetic Studies on Halipeptins, Anti-Inflammatory Cyclodepsipeptides.
Peptide Science 2005, 39-42 (2006).
176.
Kazuishi Makino, Takefumi Fujii and Yasumasa Hamada: Rhodium-Catalyzed
Asymmetric Hydrogenation through Dynamic Kinetic Resolution: Asymmetric
Synthesis of anti b-Hydroxy-a-amino Acid Esters. Tetrahedron: Asymmetry, 17,
481-485 (2006).
175.
Sousuke Hara, Kazuishi Makino, and Yasumasa Hamada: Total Synthesis of
Halipeptin A, a Potent Antiinflammatory Cyclodepsipeptide from Marine Sponge. Tetrahedron Lett., 47, 1081-1085 (2006).
174.
Osamu Hara, Taiju Nakamura, Kazuishi Makino, and Yasumasa Hamada: Synthesis of
Naphthothiazolium Salts from BINOL. Heterocycles,
68, 101-110 (2006).
173.
Osamu Hara, Taiju Nakamura, Fumihiko Sato, Kazuishi Makino, and Yasumasa
Hamada: Palladium-catalyzed Cross-coupling Reaction of 4-Methylthiazole and
2-Trimethylsilylthiazoles with Biaryl Triflates. Heterocycles 68, 1-4 (2006).
2005
172.
Tomoyuki Hasegawa, Yasufumi Kawanaka, Eichi Kasamatsu, Chisa Ohta, Kazuhiro
Nakabayashi, Masaki Okamoto, Masaya Hamano, Keiji Takahashi, Shuichi Ohuchida
and Yasumasa Hamada: A New Process for Synthesis of
the Astrocyte Activation Suppressor, ONO-2506. Org. Process Res. Dev.,
9, 774 – 781
(2005).
171.
Kazuishi Makino, Ikuko Ogawa, and Yasumasa Hamada: Synthesis of New Chiral Bis-oxazoline
Ligand with Zinc Triflate-selective Chelating Ability and Its Application to
Enantioselective Diels-Alder Cycloaddition Reaction. Heterocycles, 66,
433-440 (2005).
170.
Tetsuhiro Nemoto, Takamasa Masuda, Yuichi Akimoto, Takashi Fukuyama, and
Yasumasa Hamada: Pd-catalyzed Asymmetric Allylic Amination Using Aspartic
acid-derived P-Chirogenic Diaminophosphine Oxides: DIAPHOXs. Organic Lett., 7, 4447-4450 (2005).
169.
Kazuishi Makino, Eri Nagata, and Yasumasa Hamada: Practical Synthesis of (2S,3R)-3-Hydroxy-3-methylproline,
a Constituent of Polyoxypeptins, Using a Tandem Michael-aldol Reaction Tetrahedron Lett. 46(47)
8159-8162(2005).
168.
Kazuishi Makino, Eri Nagata, and Yasumasa Hamada: Synthesis of Tripeptide
Hydrolysate from Papuamide A – Determination of Absolute Stereostructure of b-Methoxytyrosine. Tetrahedron Lett. 46(40) 6827-6830
(2005).
167.
Tetsuhiro Nemoto, Tomoaki Fukuda, Takayoshi Matsumoto, Tsukasa Hitomi, and
Yasumasa Hamada: Enantioselective Construction of All-Carbon Quaternary
Stereocenters Using Pd-Catalyzed Asymmetric Allylic Alkylation of g-Acetoxy a,b-Unsaturated
Carbonyl Compounds. Advanced Synthesis & Catalysis 347, 1504-1506 (2005).
166.
Tetsuhiro Nemoto, Takamasa Masuda, Takayoshi Matsumoto, and Yasumasa Hamada:
Development of a New Class of Chiral Phosphorus Ligands: P-Chirogenic
Diaminophosphine Oxides. A Unique Source of Enantioselection in Pd-Catalyzed
Asymmetric Construction of Quaternary Carbons. J. Org. Chem.,70,7172-7178
(2005).
165.
Kazuishi Makino, Yasuhiro Hiroki, and Yasumasa Hamada: Dynamic Kinetic Resolution
catalyzed by Ir-Axially Chiral Phosphine Catalyst: Asymmetric Synthesis of Anti
Aromatic b-Hydroxy-a-amino Acid Esters. J. Am. Chem. Soc., 127, 5784-5785
(2005).
164.
Kazuishi Makino, Yoshiaki Henmi, Makiko Terasawa, Osamu Hara, and Yasumasa
Hamada: Remarkable Effects of Titanium Tetrachloride
in Diastereoselective Aza Diels-Alder Cycloaddition: Synthesis of (S)-Piperazic acid. Tetrahedron Lett., 46, 555-558
(2005).
163.
Taiju Nakamura, Osamu Hara, Tsutomu Tamura, Kazuishi Makino, and Yasumasa Hamada: A
Facile Synthesis of Chroman-4-ones and 2,3-Dihydroquinolin-4-ones with
Quaternary Carbon Using Intramolecular Stetter Reaction Catalyzed by Thiazolium
Salt. Synlett, 155-157 (2005).
2004
162.
Yoshiaki Henmi, Kazuishi Makino, Yayoi Yoshitomi, Osamu Hara, and Yasumasa
Hamada: Highly Efficient Synthesis of Piperazic Acids using Proline-catalyzed
Asymmetric a-Hydrazination. Tetrahedron:
Asymmetry, 15, 3477-3481 (2004).
161.
Tatsuya Suzuki, Kazuishi Makino, and Yasumasa Hamada:Synthetic Studies on Polyoxypeptins. Peptide Science 2003,
57-60 (2004).
160.
Sousuke Hara, Kazuishi Makino, Yasumasa Hamada: Stereoselective Synthesis of Protected (2S, 3S)-N-Methyl-5-hydroxyisoleucine, a
Component of Halipeptins. Tetrahedron,
60, 8031-8035 (2004).
159.
Osamu Hara, Kazuhiko Sugimoto, Kazuishi Makino, and Yasumasa Hamada: New
Synthesis of a Pyrroloquinoline Skeleton, the Martinelline Core, Using a Tandem
Michael–Aldol Strategy. Synlett, 1625-1627
(2004).
158.
Osamu Hara, Kazuhiko Sugimoto, and Yasumasa Hamada: Synthetic Studies on
Bradykinin Antagonist Martinellines: The Construction of Pyrrolo[3,2-c]quinoline
Skeleton using Allylic Amination and Silicon-tether RCM Reaction. Tetrahedron, 60, 9381-9390 (2004).
157.
Tetsuhiro Nemoto, Takayoshi Matsumoto, Takamasa Masuda, Tsukasa Hitomi,
Keiichiro Hatano, Yasumasa Hamada: P-Chirogenic Diaminophosphine Oxide: A New
Class of Chiral Phosphorous Ligands for Asymmetric Catalysis. J. Am. Chem. Soc., 126, 3690-3691 (2004).
156.
Kazuishi Makino, Tatsuya Suzuki, and Yasumasa Hamada: A Short-step Synthesis of
(2S, 3R)-3-Hydroxy-3-methylproline, a Component of Polyoxypeptins, Using Tandem
Michael-aldol Reaction and Optical Resolution. Bull. Chem. Soc. Jpn,77, 1694-1653 (2004).
155.
Kazuishi Makino, Takayuki Goto, Yasuhiro Hiroki, and Yasumasa Hamada:
Stereoselective Synthesis of Anti b-Hydroxy-a-amino Acids through Dynamic Kinetic
Resolution. Angew. Chem. Int. Ed., 43, 882-884 (2004).
2003
154.
Kazuishi Makino, Takayuki Katano, Yuko Takiguchi, Osamu Hara, and Yasumasa
Hamada: Efficient Construction of 1,2-Dihydroquinoline and
1,2,3,4-Tetrahydroquinoline Rings Using Tandem Michael-aldol Reaction. Tetrahedron Lett.,
44, 8925-8929 (2003).
153.
Pabba Chittari, Yasumasa Hamada, and Takayuki Shioiri: A
Synthetic Approach to Bengazoles: A Synthesis of Deacylbengazole. Heterocycles, 59, 465-472 (2003).
152.
Takayuki Shioiri, Shigekazu Sasaki, and Yasumasa Hamada: >Synthetic Approach to Microsclerodermins: Construction of Three
Building Blocks. ARKIVOC, 103-122
(2003).
2002
151.
Kazuishi Makino, Tatsuya Suzuki, Shinobu Awane, Osamu Hara, and Yasumasa
Hamada: Synthesis of the Acyl Side Chain Segment of Polyoxypeptins Using
Regioselective Ring-opening of Chiral 2, 3-Epoxy Alcohol. Tetrahedron Lett., 43,
9391-9395 (2002).
150.
Kazuishi Makino, Kensuke Shintani, Takahiro Yamatake, Osamu Hara, Keiichiro
Hatano, and Yasumasa Hamada: Stereoselective Synthesis of (S)-(+)-Lycoperdic Acid through an Endo Selective Hydroxylation of
the Chiral Bicyclic Lactam Enolate with MoOPH. Tetrahedron, 58,
9737-9740 (2002).
149.
Naoki Okamoto, Osamu Hara, Kazuishi Makino, and Yasumasa Hamada:
Diastereoselective Synthesis of All Stereoisomers of b-Methoxytyrosine,
a Component of Papuamides. J. Org. Chem.,
67, 9210-9215 (2002).
148.
Kazuishi Makino, Ai Kondoh, and Yasumasa Hamada: Synthetic Studies on
Polyoxypeptins: Stereoselective Synthesis of (2S, 3R)-3-Hydroxy-3-methylproline
using SmI2-mediated Cyclization Tetrahedron
Lett., 43, 4695-4698 (2002).
147.
Yasumasa Hamada, Iyo Kunimune, Osamu Hara: Asymmetric Synthesis of
Tetrahydroquinoline Derivative, A Building Block of Martinellines, via
Intramolecular Allylic Amination using 9-PBN. Heterocycles,55,
419-424 (2002).
146.
Kazuishi Makino, Yoshiaki Henmi, and Yasumasa Hamada; Synthetic Studies on a
Cyclic Hexadepsipeptide GE3: Stereoselective Construction of the Acyl Side
Chain. Synlett, 613-615 (2002).
2001
145.
Kazuishi Makino, Naoki Okamoto, Osamu Hara, and Yasumasa Hamada: Efficiently
Enantioselective Synthesis of (2R, 3R)- and (2S, 3S)-3-Hydroxyleucines
and Their Diastereomers through Dynamic Kinetic Resolution. Tetrahedron: Asymmetry, 12,
1757-1762 (2001).
144.
Naoki Okamoto, Osamu Hara, Kazuishi Makino, and Yasumasa Hamada:
Stereoselective Synthesis of (3S, 4R)-3,4-Dimethyl-(S)-glutamine and the Absolute Stereochemistry of Natural One from
Papuamides and Callipeltin. Tetrahedron:
Asymmetry, 12, 1353-1358 (2001).
143.
Takayuki Shioiri and Yasumasa Hamada: Efficient Syntheses of Biologically
Active Peptides of Aquatic Origin Involving Unusual Amino Acids. Synlett, 184-201 (2001).
142.
Yasumasa Hamada, Ken-ei Sakaguchi, Keiichiro Hatano, and
Osamu Hara: Asymmetric Allylic Substitution Reactions of 2-Substituted
2-Cycloalkenyl Carbonates using 9-PBN Coordinated Palladium. Tetrahedron
Lett., 42, 1297-1299 (2001).
141.
Osamu Hara, Kazushige Fujii, Yasumasa Hamada, and Youji
Sakagami: Synthesis of 2,5-Disubstituted Tetrahydrofurans Catalyzed by Palladium
(0). Heterocycles,54, 419-424 (2001).
2000
140.
Yasumasa Hamada，Naoki Okamoto, Osamu Hara, Synthesis of New Chiral Amines,
2,6-Dimethyl-9-azabicyclo[3.3.1]nonane and Its Derivatives.Heterocycles, 52, 929-934 (2000).
※1999年以前の論文はこちらのページからどうぞ。